Roland Baur

A GABA(A) receptor of defined subunit composition and positioning: concatenation of five subunits.

N-Substituted 4-amino-3,3-dipropyl-2(3H)-furanones: new positive allosteric modulators of the GABA(A) receptor sharing electrophysiological properties with the anticonvulsant loreclezole.

Functional characterization of the new human GABA(A) receptor mutation beta3(R192H).

Forced subunit assembly in alpha1beta2gamma2 GABAA receptors. Insight into the absolute arrangement.

Anxiolytic effect of wogonin, a benzodiazepine receptor ligand isolated from Scutellaria baicalensis Georgi.

On high- and low-affinity agonist sites in GABAA receptors.

Naturally occurring 2'-hydroxyl-substituted flavonoids as high-affinity benzodiazepine site ligands.

Individual properties of the two functional agonist sites in GABA(A) receptors.

The flavone hispidulin, a benzodiazepine receptor ligand with positive allosteric properties, traverses the blood-brain barrier and exhibits anticonvulsive effects.

Benzodiazepines affect channel opening of GABA A receptors induced by either agonist binding site.

Conformational changes at benzodiazepine binding sites of GABA(A) receptors detected with a novel technique.

Novel plant substances acting as beta subunit isoform-selective positive allosteric modulators of GABAA receptors.

Homeopathic medical practice: long-term results of a cohort study with 3981 patients.

Influence of the point mutation alpha-1-H101R on the assembly of gamma-aminobutyric acid type A receptors.

Consequence of the presence of two different beta subunit isoforms in a GABA(A) receptor.

Proximity-accelerated chemical coupling reaction in the benzodiazepine-binding site of gamma-aminobutyric acid type A receptors: superposition of different allosteric modulators.

Two neighboring residues of loop A of the alpha1 subunit point towards the benzodiazepine binding site of GABAA receptors.

Replacement of histidine in position 105 in the α₅ subunit by cysteine stimulates zolpidem sensitivity of α₅β₂γ₂ GABA(A) receptors.

The promiscuous role of the epsilon subunit in GABAA receptor biogenesis.

Novel chloride channel mutations leading to mild myotonia among Chinese.

Covalent modification of GABAA receptor isoforms by a diazepam analogue provides evidence for a novel benzodiazepine binding site that prevents modulation by these drugs.

Unanticipated structural and functional properties of delta-subunit-containing GABAA receptors.

Homeopathic treatment of patients with chronic low back pain: A prospective observational study with 2 years' follow-up.

Structure of alpha6 beta3 delta GABA(A) receptors and their lack of ethanol sensitivity.

Relative positioning of diazepam in the benzodiazepine-binding-pocket of GABA receptors.

Use of concatamers to study GABAA receptor architecture and function: application to delta-subunit-containing receptors and possible pitfalls.

Highly potent modulation of GABA(A) receptors by valerenic acid derivatives.

Diversity of structure and function of alpha1alpha6beta3delta GABAA receptors: comparison with alpha1beta3delta and alpha6beta3delta receptors.

Monepantel allosterically activates DEG-3/DES-2 channels of the gastrointestinal nematode Haemonchus contortus.

A residue close to α1 loop F disrupts modulation of GABAA receptors by benzodiazepines while their binding is maintained.

The major central endocannabinoid directly acts at GABA(A) receptors.

Influence of GABA(A) receptor α subunit isoforms on the benzodiazepine binding site.

Molecular analysis of the site for 2-arachidonylglycerol (2-AG) on the β₂ subunit of GABA(A) receptors.

Effects and feasibility of an Integrative Medicine program for geriatric patients-a cluster-randomized pilot study.

acr-23 Encodes a monepantel-sensitive channel in Caenorhabditis elegans.

Dementia: treating patients and caregivers with complementary and alternative medicine--results of a clinical expert conference using the World Café method.

Do N-arachidonyl-glycine (NA-glycine) and 2-arachidonoyl glycerol (2-AG) share mode of action and the binding site on the β2 subunit of GABAA receptors?

Accelerated discovery of novel benzodiazepine ligands by experiment-guided virtual screening.

Moderate concentrations of 4-O-methylhonokiol potentiate GABAA receptor currents stronger than honokiol.

A pentasymmetric open channel blocker for Cys-loop receptor channels.

Monepantel irreversibly binds to and opens Haemonchus contortus MPTL-1 and Caenorhabditis elegans ACR-20 receptors.

Structural analogues of the natural products magnolol and honokiol as potent allosteric potentiators of GABA(A) receptors.

Positive modulation of synaptic and extrasynaptic GABAA receptors by an antagonist of the high affinity benzodiazepine binding site.

Modulatory Effects of Eschscholzia californica Alkaloids on Recombinant GABAA Receptors.

Functional sites involved in modulation of the GABAA receptor channel by the intravenous anesthetics propofol, etomidate and pentobarbital.

A new chromanone derivative isolated from Hypericum lissophloeus (Hypericaceae) potentiates GABAA receptor currents in a subunit specific fashion.

Novel positive allosteric modulators of GABAA receptors with anesthetic activity.

Molecular mode of action of CGS 9895 at α1 β2 γ2 GABAA receptors.

Toward Understanding Functional Properties and Subunit Arrangement of α4β2δ γ-Aminobutyric Acid, Type A (GABAA) Receptors.