Ralf Schirrmacher

¹⁸F-labeled silicon-based fluoride acceptors: potential opportunities for novel positron emitting radiopharmaceuticals.

5-(4-((4-[(18)F]Fluorobenzyl)oxy)-3-methoxybenzyl)pyrimidine-2,4-diamine: a selective dual inhibitor for potential PET imaging of Trk/CSF-1R.

In Vivo Evaluation of ¹⁸F-SiFAlin-Modified TATE: A Potential Challenge for ⁶⁸Ga-DOTATATE, the Clinical Gold Standard for Somatostatin Receptor Imaging with PET.

Improving the stability of peptidic radiotracers by the introduction of artificial scaffolds: which structure element is most useful?

Evaluation of WO2015042088 A1 - a novel urea-based scaffold for TrkA inhibition.

From Unorthodox to Established: The Current Status of (18)F-Trifluoroborate- and (18)F-SiFA-Based Radiopharmaceuticals in PET Nuclear Imaging.

Recent Advances in the Development and Application of Radiolabeled Kinase Inhibitors for PET Imaging.

Radiosynthesis and Preclinical Evaluation of F-Fluoroglycosylated Octreotate for Somatostatin Receptor Imaging.

Tropomyosin receptor kinase inhibitors: an updated patent review for 2010-2016 - Part I.

Tropomyosin receptor kinase inhibitors: an updated patent review for 2010-2016 - Part II.

Design and synthesis of a fluorinated quinazoline-based type-II Trk inhibitor as a scaffold for PET radiotracer development.

A Kinome-Wide Selective Radiolabeled TrkB/C Inhibitor for in Vitro and in Vivo Neuroimaging: Synthesis, Preclinical Evaluation, and First-in-Human.

Small Prosthetic Groups in F-Radiochemistry: Useful Auxiliaries for the Design of F-PET Tracers.

Automated synthesis of PET radiotracers by copper-mediated F-fluorination of organoborons: Importance of the order of addition and competing protodeborylation.

Synthesis, in vitro and in vivo evaluation of F-fluoronorimatinib as radiotracer for Imatinib-sensitive gastrointestinal stromal tumors.

F-Radiolabeling and In Vivo Analysis of SiFA-Derivatized Polymeric Core-Shell Nanoparticles.

Identification of [F]TRACK, a Fluorine-18-Labeled Tropomyosin Receptor Kinase (Trk) Inhibitor for PET Imaging.

Recent Advances in F Radiochemistry: A Focus on B-F, Si-F, Al-F, and C-F Radiofluorination via Spirocyclic Iodonium Ylides.

Gastrin-Releasing Peptide Receptor- and Prostate-Specific Membrane Antigen-Specific Ultrasmall Gold Nanoparticles for Characterization and Diagnosis of Prostate Carcinoma via Fluorescence Imaging.

Design, synthesis and in vitro evaluation of heterobivalent peptidic radioligands targeting both GRP- and VPAC-Receptors concomitantly overexpressed on various malignancies - Is the concept feasible?

Design, Synthesis, In Vitro, and Initial In Vivo Evaluation of Heterobivalent Peptidic Ligands Targeting Both NPY(Y₁)- and GRP-Receptors-An Improvement for Breast Cancer Imaging?

iEDDA Conjugation Reaction in Radiometal Labeling of Peptides with Ga and Cu: Unexpected Findings.

Radioligands for Tropomyosin Receptor Kinase (Trk) Positron Emission Tomography Imaging.

First-in-Human Brain Imaging of [F]TRACK, a PET tracer for Tropomyosin Receptor Kinases.