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Chapter 6

Drugs Acting on Autonomic Nervous System: Adrenergic Agonists and Antagonists Agents

Neuronas Adrenúdicas: Neurotransmisión
Neuronas Adrenúdicas: Neurotransmisión
Postganglionic sympathetic fibers (except those supplying the sweat glands) releasing noradrenaline or norepinephrine are called noradrenergic or ...
Receptores Adrenérgicos (Adrenoceptores): Clasificación
Receptores Adrenérgicos (Adrenoceptores): Clasificación
Adrenergic receptors, or adrenoceptors, respond to the autonomic neurotransmitter noradrenaline and other endogenous catecholamine agonists. They are ...
Receptores adrenérgicos: ɑ Subtipo
Receptores adrenérgicos: ɑ Subtipo
Adrenoceptors are classified into α and ꞵ classes based on their potencies to catecholamine agonists. α-adrenoceptors show the following ...
Receptores adrenérgicos: subtipo β
Receptores adrenérgicos: subtipo β
β-adrenoceptors have varied sensitivities towards adrenaline, noradrenaline, and isoprenaline. The order of agonist potency is as follows: ...
Agonistas adrenérgicos: agentes de acción directa
Agonistas adrenérgicos: agentes de acción directa
Drugs that mimic the action of endogenous catecholamines like noradrenaline and adrenaline are called adrenergic agonists or sympathomimetics. Based on ...
Agonistas adrenérgicos: agentes de acción indirecta
Agonistas adrenérgicos: agentes de acción indirecta
Indirect-acting adrenergic agonists potentiate the effects of endogenous catecholamines through different mechanisms without directly binding to ...
Agonistas adrenérgicos: agentes de acción mixta
Agonistas adrenérgicos: agentes de acción mixta
Mixed-action adrenergic agonists, like ephedrine and pseudoephedrine, directly and indirectly affect adrenergic receptors. These agents stimulate ...
Agonistas adrenérgicos: química y relación estructura-actividad
Agonistas adrenérgicos: química y relación estructura-actividad
Adrenergic agonists' structure-activity relationship (SAR) determines their selectivity and efficacy. These agonists comprise a phenylethylamine ...
Agonistas adrenérgicos: clasificación terapéutica
Agonistas adrenérgicos: clasificación terapéutica
Adrenergic agonists can be classified based on their therapeutic uses and mechanisms of action. They serve various purposes in clinical applications. ...
Agonistas adrenérgicos: usos terapéuticos
Agonistas adrenérgicos: usos terapéuticos
Adrenergic agonists have diverse therapeutic uses across various medical conditions and emergencies. Emergency and Intensive Care Unit (ICU) applications: ...
Antagonistas adrenérgicos: química y clasificación de los bloqueadores de los receptores ɑ
Antagonistas adrenérgicos: química y clasificación de los bloqueadores de los receptores ɑ
Adrenergic antagonists, or sympatholytics, inhibit adrenoceptor activation driven by catecholamines or agonists. Based on their adrenoceptor specificity, ...
Antagonistas Adrenérgicos: Acciones Farmacológicas de los Bloqueadores de los Receptores ɑ
Antagonistas Adrenérgicos: Acciones Farmacológicas de los Bloqueadores de los Receptores ɑ
α-Adrenergic antagonists, known as α-blockers, exert their effects by inhibiting α-adrenoceptors, leading to specific physiological ...
Antagonistas adrenérgicos: química y clasificación de los bloqueadores de los receptores de β
Antagonistas adrenérgicos: química y clasificación de los bloqueadores de los receptores de β
β-adrenergic antagonists, or β-blockers, modulate the sympathetic nervous system by targeting β-adrenoceptors and inhibiting ...
Antagonistas Adrenérgicos: Acciones Farmacológicas de los Bloqueadores de los Receptores β
Antagonistas Adrenérgicos: Acciones Farmacológicas de los Bloqueadores de los Receptores β
β-receptor blockers significantly impact the cardiovascular system by counteracting catecholamine-induced sympathetic responses. These medications ...
Antagonistas adrenérgicos: bloqueadores de los receptores ɑ y β
Antagonistas adrenérgicos: bloqueadores de los receptores ɑ y β
Third-generation β-blockers, such as labetalol and carvedilol, represent a significant advancement in managing cardiovascular conditions. Unlike ...
Fármacos que afectan a la síntesis de neurotransmisores
Fármacos que afectan a la síntesis de neurotransmisores
Drugs affecting neurotransmitter synthesis can impact the adrenergic neuron and the synthesis of neurotransmitters. For example, α-methyltyrosine and ...
Fármacos que afectan a la liberación o absorción de neurotransmisores
Fármacos que afectan a la liberación o absorción de neurotransmisores
Certain drugs can affect how neurotransmitters called catecholamines, are released or taken back up in the adrenergic neuron. They can have different ...
Glaucoma: Información general
Glaucoma: Información general
Glaucoma is an eye condition characterized by increased intraocular pressure that damages the retina and optic nerve, leading to irreversible blindness if ...
Glaucoma de ángulo abierto: tratamiento
Glaucoma de ángulo abierto: tratamiento
In open-angle glaucoma, the iridocorneal angle remains open, but the trabecular meshwork becomes stiff, slowing down the outflow of aqueous humor. This ...
Glaucoma con cierre de ángulo: tratamiento
Glaucoma con cierre de ángulo: tratamiento
Angle-closure glaucoma, or closed-angle glaucoma, is an eye condition where the iris bulges out and blocks the iridocorneal angle, resulting in a buildup ...
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