Results: Representative Target Engagement Quantification by High Content Imaging
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Conclusion
副本
This method can help answer key questions in chemical biology and drug discovery. Such as, does your compound bind to the target protein? The main advantages for this technique are that there's no requirement of detachment of the adherent cells.</
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Measurements of drug target engagement are central to effective drug development and chemical probe validation. Here, we detail a protocol for measuring drug-target engagement using high content imaging in a microplate-compatible adaption of the cellular thermal shift assay (CETSA).